题名 | Discovery of 1-{4-[3-Fluoro-4-((3S,6R)-3-methyl-1,1-dioxo-6-phenyl-[1,2]thiazinan-2-ylmethyl)-phenyl]-piperazin-1-yl}-ethanone (GNE-3500): a Potent, Selective, and Orally Bioavailable Retinoic Acid Receptor-Related Orphan Receptor C (RORc or RORγ) Inverse Agonist. |
杂志 | J Med Chem. 2015 Jun 10 |
链接 | http://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.5b00597 |
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